產(chǎn)品名稱 LDC 000067 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 6752/5
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameLDC 000067
DescriptionPotent and selective CDK9 inhibitor (IC50 = 44 nM at CDK9-cyclin T1). Inhibits other CDKs in the micromolar range (IC50 values are 2.4, 5.5, 9.2, >10 and >10 μM for CDK2-cyclin A, CDK1-cyclin B1, CDK4-cyclin D1, CDK6-cyclin D3 and CDK7-cyclin H-MAT1, respectively). Inhibits P-TEFb-dependent in vitro transcription. Induces apoptosis in vitro and in vivo in combination with BI 894999. Purity 98%. MW (observed): 370.43
Size5 mg
Concentrationn/a
Applicationsn/a
Other Names3-[[6-(2-Methoxyphenyl)-4-pyrimidinyl]amino]benzenemethanesulfonamide
Gene, Accession, CAS #CAS: 1073485-20-7
Catalog #6752/5
Price
Order / More InfoLDC 000067 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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