產(chǎn)品名稱 BIX 01294 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 3364/10
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameBIX 01294
DescriptionGLP and G9a histone lysine methyltransferase inhibitor (IC50 values are 0.7 and 1.7 μM respectively) that displays no activity at other histone methyltransferases up to 37 μM. Modulates H3K9me2 levels in mammalian cells and potentiates induction of pluripotent stem cells from somatic cells in vitro. Also inhibits H3K36 methylation by oncoproteins NSD1, NSD2 and NSD3 (IC50 values are 40 - 112 μM). Purity 98%. MW (observed): 600.02
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names2-(Hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6,7-dimethoxy-N-[1-(phenylmethyl)-4-piperidinyl]-4-quinazolinamine trihydrochloride
Gene, Accession, CAS #CAS: 1392399-03-9
Catalog #3364/10
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Order / More InfoBIX 01294 from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 21209933
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