產(chǎn)品名稱 BIX-01294 from ARBOR ASSAYS, INC.
產(chǎn)品貨號 P018-25MG
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 25 mg
產(chǎn)品品牌 ARBOR ASSAYS, INC.
產(chǎn)品概述
產(chǎn)品詳情
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Product NameBIX-01294
DescriptionBIX-01294, a diazepin-quinazolinamine derivative, is a selective,cell-permeable G9a-like protein and G9a histone lysine methyltransferase (HMTase) inhibitor (IC50 values are 0.7 and 1.7 uM respectively) that displays little or no activity at other HMTases. BIX-01294 has been used in combination with the calcium channel activator BayK8644 to facilitate the generation of induced pluripotent stem cells from somatic cells in vitro. BIX-01294 and valproic acid, a histone deacetylase (HDAC) inhibitor, may replace the requirement for ectopic OCT4 (POU5F1) and cMyc respectively in pluripotent stem cell induction (iPS) recipes.
Size25 mg
Concentrationn/a
ApplicationsActivator or Inhibitor
Other NamesHMT inhibitor
Gene, Accession, CAS #n/a
Catalog #P018-25MG
Price
Order / More InfoBIX-01294 from ARBOR ASSAYS, INC.
Product Specific Referencesn/a
產(chǎn)品資料
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