| 產(chǎn)品詳情 |
| Edit |   |
|---|
| Product Name | INCB 3284 dimesylate |
|---|
| Description | Potent, selective hCCR2 antagonist. Exhibits potent antagonism against monocyte chemoattractant molecule binding to hCCR2 and chemotaxis activity (IC50 values are 3.7 and 4.7 nM respectively). Also displays weak hERG activity; inhibits the hERG potassium current (IC50 = 84μM). Orally bioavailable. Purity 98%. MW (observed): 712.76 |
|---|
| Size | 50 mg |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | N-[2-[[(3R)-1-[trans-4-Hydroxy-4-(6-methoxy-3-pyridinyl)cyclohexyl]-3-pyrrolidinyl]amino]-2-oxoethyl]-3-(trifluoromethyl)-benzamide dimethanesulfonate |
|---|
| Gene, Accession, CAS # | CAS: 887401-93-6 |
|---|
| Catalog # | 4306/50 |
|---|
| Price | |
|---|
| Order / More Info | INCB 3284 dimesylate from TOCRIS BIOSCIENCE
|
|---|
| Product Specific References | PubMed: 24904083, 25012628, 27216982 |
|---|
| 產(chǎn)品資料 |
|
|