產(chǎn)品名稱 LY 344864 hydrochloride from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 2451/50
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameLY 344864 hydrochloride
DescriptionPotent, selective 5-HT1F receptor agonist (EC50 = 3 nM). Displays > 80-fold selectivity over other 5-HT receptors (Ki values are 0.006, 0.53, 0.55, 0.56, 1.42, 1.70, 3.50, 3.94 and 4.85 μM for 5-HT1F, 5-HT1A, 5-HT1B, 5-HT1D, 5-HT1E, 5-HT2B, 5-HT2C, 5-HT2A and 5-HT7 receptors respectively). Inhibits neurogenic dural inflammation in vivo following i.v. and oral administration. Purity 99%. MW (observed): 387.88
Size50 mg
Concentrationn/a
Applicationsn/a
Other NamesN-[(3R)-3-(Dimethylamino)-2,3,4,9-tetrahydro-1H-carbazol-6-yl]-4-fluorobenzamide hydrochloride
Gene, Accession, CAS #CAS: 1217756-94-9
Catalog #2451/50
Price
Order / More InfoLY 344864 hydrochloride from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 21653728, 24849926
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