產(chǎn)品名稱 SEN 12333 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 4441/50
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameSEN 12333
Descriptionα7 nicotinic acetylcholine receptor (nAChR) agonist (EC50 = 1.6 μM, Ki = 260 nM at rat α7 nAChRs). Also displays functional antagonism at histamine H3 receptors (IC50 = 103 nM) and weak agonist activity at human ganglionic α3 nAChRs (IC50 = 8.5 μM). Neuroprotective in a rodent model of quisqualic acid-induced cholinergic degeneration. Brain penetrant and orally bioavailable. Purity 99%. MW (observed): 339.43
Size50 mg
Concentrationn/a
Applicationsn/a
Other NamesN-[4-(3-pyridinyl)phenyl]-4-morpholinepentanamide. WAY 317538
Gene, Accession, CAS #CAS: 874450-44-9
Catalog #4441/50
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Order / More InfoSEN 12333 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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