產品名稱 DREADD agonist 21 from TOCRIS BIOSCIENCE
產品貨號 5548/50
產品價格 現(xiàn)貨詢價,電話:010-67529703
產品規(guī)格 50 mg
產品品牌 TOCRIS BIOSCIENCE
產品概述
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Product NameDREADD agonist 21
DescriptionPotent muscarinic DREADD agonist (pEC50 values are 8.91, 8.48 and 7.77 for hM1Dq, hM3Dq and hM4Di in vitro, respectively). Exhibits > 10-fold higher affinity for hM1Dq and hM4Di compared to wild type receptors. Also displays little to no activity at wild type M3 receptors. Activates neurons expressing hM3Dq DREADDS and inhibits activity in neurons expressing hM4Di in vivo. Displays excellent brain permeability. Water soluble salt also available, DREADD agonist 21 hydrochloride (Cat. No. 6422). Purity 98%. MW (observed): 278.35
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names11-(1-Piperazinyl)-5H-dibenzo[b,e][1,4]diazepine
Gene, Accession, CAS #CAS: 56296-18-5
Catalog #5548/50
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Order / More InfoDREADD agonist 21 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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