產(chǎn)品名稱 PF 915275 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 3291/50
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NamePF 915275
DescriptionPotent and selective 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1) inhibitor (Ki = 2.3 nM) that displays little activity at 11βHSD2 (1.5% inhibition at 10 μM). Inhibits the conversion of prednisone to prednisolone in human hepatocytes in vitro (EC50 = 15 nM) and has antidiabetic activity in vivo. Orally active. Purity 98%. MW (observed): 350.39
Size50 mg
Concentrationn/a
Applicationsn/a
Other NamesN-(6-Amino-2-pyridinyl)-4'-cyano-[1,1'-biphenyl]-4-sulfonamide
Gene, Accession, CAS #CAS: 857290-04-1
Catalog #3291/50
Price
Order / More InfoPF 915275 from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 23927023, 30021644
產(chǎn)品資料
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