產(chǎn)品名稱(chēng) PF 06424439 from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 6348/5
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NamePF 06424439
DescriptionPotent and selective DGAT2 inhibitor (IC50 = 14 nM). Exhibits no significant activity at MGAT1-3 or DGAT1. Reduces triglyderide synthesis in human hepatocytes in vitro. Reduces plasma triglyceride and cholesterol levels in a rat dyslipidemia model. Orally bioavailable. Purity 98%. MW (observed): 536.05
Size5 mg
Concentrationn/a
Applicationsn/a
Other Names[(3R)-1-[2-[1-(4-Chloro-1H-pyrazol-1-yl)cyclopropyl]-3H-imidazo[4,5-b]pyridin-5-yl]-3-piperidinyl]-1-pyrrolidinylmethanone methanesulfonate
Gene, Accession, CAS #CAS: 1469284-79-4
Catalog #6348/5
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Order / More InfoPF 06424439 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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