產(chǎn)品名稱 CP 724714 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 5973/10
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameCP 724714
DescriptionPotent and selective ErbB2 inhibitor (IC50 = 10 nM). Exhibits 500-1000-fold selectivity for ErbB2 over ErbB1 and other related RTKs. Induces G1 cell cycle arrest in an ErbB2-overexpressing human cancer cell line. Promotes tumor apoptosis. Induces tumor regression in a human tumor xenograft model. Displays no apparent toxic effect on cardiac tissue. Purity 98%. MW (observed): 469.53
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names2-Methoxy-N-[(2E)-3-[4-[[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]phenyl]amino]-6-quinazolinyl]-2-propen-1-yl]acetamide
Gene, Accession, CAS #CAS: 383432-38-0
Catalog #5973/10
Price
Order / More InfoCP 724714 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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