產(chǎn)品名稱 Methoctramine from CAYMAN CHEMICAL COMPANY
產(chǎn)品貨號 24317-10
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
產(chǎn)品概述
產(chǎn)品詳情
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Product NameMethoctramine
DescriptionA selective muscarinic M2 receptor antagonist (IC50 = 6.1 nM in CHO-K1 cell membranes); selective for M2 over M1, M3, M4, and M5 receptors (IC50s = 92, 770, 260, and 217 nM, respectively); inhibits acetylcholine-induced reductions in isolated guinea pig tracheal tube contractions in vitro (1 μM); inhibits bradycardia and bronchoconstriction induced by acetylcholine in guinea pigs (ED50s = 38 and 81 nmol/kg, respectively); suppresses oxotremorine M-induced bladder overactivity in a rat model of spinal cord injury
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names104807-40-1 M-2 1 3 4 5 CHOK1
Gene, Accession, CAS #CAS: 104807-46-7
Catalog #24317-10
Price
Order / More InfoMethoctramine from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
產(chǎn)品資料
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