| 產(chǎn)品詳情 |
| Edit |   |
|---|
| Product Name | Cortistatin-14 (trifluoroacetate salt) |
|---|
| Description | An endogenous neuropeptide agonist of SST1-SST5 (IC50s = 0.5-18.2 nM for human receptors expressed in CCL39 cells); [KC1] competitively inhibits hexarelin binding to GHS-R in pituitary membranes (Ki = 0.54 μM); activates the human MrgX2 receptor expressed in HEK293 cells (EC50 = 1.3 μM); completely inhibits TRH, and partially inhibits VIP, stimulation of cAMP production in GH4 cells (0.01-1 μM); dose-dependently impairs memory retention in mice when delivered after foot shock avoidance training (0.05-5 μg, i.c.v.); dose-dependently reduces growth hormone secretion in rats with a reduction of over 80% at all concentrations after 10 minutes (40-320 μg/kg s.c.) |
|---|
| Size | 500 μg |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | 186901-48-4 193829-96-8 937031-00-0 CCL 39 SST GHSR GH-4 Mrg-X2 |
|---|
| Gene, Accession, CAS # | n/a |
|---|
| Catalog # | 25074-500 |
|---|
| Price | |
|---|
| Order / More Info | Cortistatin-14 (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY |
|---|
| Product Specific References | n/a |
|---|
| 產(chǎn)品資料 |
|
|