產(chǎn)品名稱(chēng) GSK 343 from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 6128/50
產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameGSK 343
DescriptionPotent and selective SAM-competitive EZH2 inhibitor (IC50 = 4 nM). Exhibits >60 fold selectivity for EZH2 over EZH1 and a range of other methyltransferases. Decreases H3K27me3 levels in breast cancer cells in vitro. Inhibits proliferation of prostate cancer cell lines in vitro. Purity 98%. MW (observed): 541.69
Size50 mg
Concentrationn/a
Applicationsn/a
Other NamesN-[(1,2-Dihydro-6-methyl-2-oxo-4-propyl-3-pyridinyl)methyl]-1-(1-methylethyl)-6-[2-(4-methyl-1-piperazinyl)-4-pyridinyl]-1H-indazole-4-carboxamide
Gene, Accession, CAS #CAS: 1346704-33-3
Catalog #6128/50
Price
Order / More InfoGSK 343 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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