產(chǎn)品名稱 GSK 269962 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 4009/50
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameGSK 269962
DescriptionPotent Rho kinase (ROCK) inhibitor (IC50 values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively). Displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases. Induces vasorelaxation in preconstricted rat aorta (IC50 = 35 nM); lowers blood pressure in a rat model of hypertension. Purity 99%. MW (observed): 570.6
Size50 mg
Concentrationn/a
Applicationsn/a
Other NamesN-[3-[[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy]phenyl]-4-[2-(4-morpholinyl)ethoxy]benzamide
Gene, Accession, CAS #CAS: 850664-21-0
Catalog #4009/50
Price
Order / More InfoGSK 269962 from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 24076962, 25261469, 25264362, 27036020, 27820945
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