產(chǎn)品名稱 LY 393558 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 3350/10
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameLY 393558
DescriptionDual 5-HT1B/1D receptor antagonist (pKB values are 9.05 and 8.98 respectively) and 5-HT re-uptake inhibitor (pIC50 = 8.48). Potently antagonizes terminal autoreceptor activity in vitro and increases extracellular 5-HT levels above those evoked by fluoxetine (Cat. No. 0927) in vivo. Also acts as an antagonist at 5-HT2A and 5-HT2B receptors (pKi values are 7.29 and 7.35 respectively). Purity 97%. MW (observed): 546.68
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names1-[2-[4-(6-Fluoro-1H-indol-3-yl)-3,6-dihydro-1(2H)-pyridinyl]ethyl]-3,4-dihydro-3-(1-methylethyl)-6-(methylsulfonyl)-1H-2,1,3-benzothiadiazine-2,2-dioxide
Gene, Accession, CAS #CAS: 271780-64-4
Catalog #3350/10
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Order / More InfoLY 393558 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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