產(chǎn)品名稱 (R)-PFI 2 hydrochloride from TOCRIS BIOSCIENCE
產(chǎn)品貨號 4892/10
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
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Product Name(R)-PFI 2 hydrochloride
DescriptionPotent and selective SETD7 histone lysine methyltransferase inhibitor (IC50 = 2 nM). Exhibits >1000-fold selectivity over DNMT1 and a panel of 18 other methyltransferases. Inhibits YAP nuclear translocation and function following activation of the Hippo signaling pathway in MCF7 cells. Negative Control also available.. Purity 97%. MW (observed): 535.98
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names(1R)-1-[[3-(Trifluoromethyl)phenyl]methyl]-2-oxo-2-(1-pyrrolidinyl)ethyl]1,2,3,4-tetrahydro-6-isoquinolinesulfonamide hydrochloride
Gene, Accession, CAS #CAS: 1627607-87-7
Catalog #4892/10
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Order / More Info(R)-PFI 2 hydrochloride from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 25136132, 25897119, 29395054
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