產(chǎn)品名稱 NVP 2 from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 6535/5
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameNVP 2
DescriptionPotent and selective ATP-competitive CDK9 inhibitor (IC50 = 0.5 nM). Exhibits selectivity for CDK9 over a panel of 468 kinases, but inhibits DYRK1B (IC50 = 350 nM), displays <90% binding to CDK7 (IC50 >10 μM) and CDK13. Inhibits proliferation of MOLT4 cells in vitro. Induces apoptosis. Purity 97%. MW (observed): 513.07
Size5 mg
Concentrationn/a
Applicationsn/a
Other Names4-[[[5'-Chloro-2'-[[trans-4-[[(1R)-2-methoxy-1-methylethyl]amino]cyclohexyl]amino][2,4'-bipyridin]-6-yl]amino]methyl]tetrahydro-2H-pyran-4-carbonitrile
Gene, Accession, CAS #CAS: 1263373-43-8
Catalog #6535/5
Price
Order / More InfoNVP 2 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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