產(chǎn)品名稱 JNJ 16259685 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 2333/10
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameJNJ 16259685
DescriptionSub-nanomolar potent, non-competitive mGlu1 antagonist (Ki = 0.34 nM). Inhibits glutamate-induced Ca2+ response at the human mGlu1 receptor with an IC50 value of 0.55 nM. Selective over mGlu5 (> 400-fold) and displays no activity at mGlu2, mGlu3, mGlu4, mGlu6, AMPA or NMDA receptors (IC50 > 10 μM). Centrally active following systemic administration. Purity 98%. MW (observed): 325.41
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names(3,4-Dihydro-2H-pyrano[2,3-b]quinolin-7-yl)-(cis-4-methoxycyclohexyl)-methanone
Gene, Accession, CAS #CAS: 409345-29-5
Catalog #2333/10
Price
Order / More InfoJNJ 16259685 from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 17502847, 18174329, 19657020, 21753005, 24205371, 24270186, 24467847, 26269634, 26655894, 27807163
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