產(chǎn)品名稱 AM 281 from TOCRIS BIOSCIENCE
產(chǎn)品貨號 1115/10
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
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Product NameAM 281
DescriptionPotent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (Ki = 14 nM). Purity 99%. MW (observed): 557.22
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide
Gene, Accession, CAS #CAS: 202463-68-1
Catalog #1115/10
Price
Order / More InfoAM 281 from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 11030713, 11877326, 12578907, 15238431, 15277316, 15564588, 15669919, 16434616, 16760924, 17234582, 17267577, 17301239, 17384130, 17408433, 17434980, 17660390, 17678736, 18156315, 19091987, 19506935, 20074214, 20136841, 20430875, 20531936, 20534730, 20590572, 21048703, 21440630, 23151067, 23152849, 23673278, 25655433, 25768340, 27424778, 28322749, 28495606, 28779174
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