產(chǎn)品名稱 Bisindolylmaleimide II from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 4128/50
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameBisindolylmaleimide II
DescriptionPotent, ATP-competitive protein kinase C (PKC) inhibitor (IC50 = 0.01 μM). Displays selectivity for PKC over protein kinase A (PKA) and phosphorylase kinase (PK) (IC50 values are 0.75 and 2μM for PK and PKA respectively). Also displays potent, noncompetitive antagonism at nicotinic cholinergic receptors (IC50 ~ 0.03 μM for inhibition of catecholamine secretion in nicotine-stimulated PC-12 cells). Purity 97%. MW (observed): 438.52
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names3-(1H-Indol-3-yl)-4-[1-[2-(1-methyl-2-pyrrolidinyl)ethyl]-1H-indol-3-yl]-1H-pyrrole-2,5-dione
Gene, Accession, CAS #CAS: 137592-45-1
Catalog #4128/50
Price
Order / More InfoBisindolylmaleimide II from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 15269224
產(chǎn)品資料
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