產(chǎn)品名稱 CPI-637 from CAYMAN CHEMICAL COMPANY
產(chǎn)品貨號 23500-5
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
產(chǎn)品概述
產(chǎn)品詳情
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Product NameCPI-637
DescriptionAn inhibitor of CBP/EP300 bromodomains (IC50s = 30 and 51 nM in a TR-FRET assay); selective for CBP and EP300 over the BET family of bromodomains (IC50s = >10 μM); is active at bromodomain BRD9 (IC50 = 0.73 μM); inhibits CBP (IC50 = 0.3 μM in a BRET assay) and inhibits MYC expression (EC50 = 0.6 μM) in AMO-1 cells
Size5 mg
Concentrationn/a
Applicationsn/a
Other NamesCPI637 fluorescence resonance energy transfer cAMP EP-300 TRFRET BRD-9 AMO1
Gene, Accession, CAS #CAS: 1884712-47-3
Catalog #23500-5
Price
Order / More InfoCPI-637 from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
產(chǎn)品資料
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