產(chǎn)品名稱 L Moses dihydrochloride from TOCRIS BIOSCIENCE
產(chǎn)品貨號 6251/50
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 50 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameL Moses dihydrochloride
DescriptionHigh affinity and selective cell-permeable p300/CBP-associated factor (PCAF) inhibitor (Ki = 47 nM). Exhibits no significant activity against a panel of 48 other bromodomains except GCN5 (Kd = 600 nM). Exhibits >4500-fold selectivity for PCAF over BRD4. Also exhibits metabolic stability in mouse and human liver microsomes and no observable cytotoxicity in peripheral blood mononuclear cells (PBMC). Purity 98%. MW (observed): 433.38
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names(1S, 2S)-N1,N1-Dimethyl-N2-(3-methyl-1,2,4-triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diamine dihydrochloride
Gene, Accession, CAS #n/a
Catalog #6251/50
Price
Order / More InfoL Moses dihydrochloride from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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