產(chǎn)品名稱 Talabostat mesylate from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 3719/10
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameTalabostat mesylate
DescriptionPotent DPP IV inhibitor (IC50 values are <4, 4, 11, 310 and 560 nM at DPP4, DPP8, DPP9, DPP7 and FAP, respectively). Activates the inflammasome sensor protein NLRP1b and selectively triggers pyroptosis in monocytes and macrophages. Induces immune-mediated tumor regression in multiple mouse models of cancer. Orally bioavailable. Purity 98%. MW (observed): 310.18
Size10 mg
Concentrationn/a
Applicationsn/a
Other NamesB-[(2R)-1-[(2S)-2-Amino-3-methyl-1-oxobutyl]-2-pyrrolidinyl]boronic acid methanesulfonate. Val-boroPro, BXCL 701
Gene, Accession, CAS #CAS: 150080-09-4
Catalog #3719/10
Price
Order / More InfoTalabostat mesylate from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 27820798
產(chǎn)品資料
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