| 產品詳情 |
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| Product Name | UNC 0642 |
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| Description | Potent and selective G9a and GLP histone lysine methyltransferase inhibitor (IC50 < 2.5 nM). Exhibits >2,000-fold selectivity for G9a and GLP over PRC2-EZH2 and >20,000-fold selectivity over other methyltransferases. Reduces H3K9 dimethylation levels in MDA-MB-231 cells (IC50 = 110 nM). Displays modest brain penetration in vivo. Purity 99%. MW (observed): 546.7 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 2-(4,4-Difluoro-1-piperidinyl)-6-methoxy-N-[1-(1-methylethyl)-4-piperidinyl]-7-[3-(1-pyrrolidinyl)propoxy]-4-quinazolinamine |
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| Gene, Accession, CAS # | CAS: 1481677-78-4 |
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| Catalog # | 5132/10 |
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| Price | |
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| Order / More Info | UNC 0642 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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| 產品資料 |
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