產(chǎn)品名稱 GSK343 from BIOVISION, INC.
產(chǎn)品貨號 2281-5
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 BIOVISION, INC.
產(chǎn)品概述
產(chǎn)品詳情
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Product NameGSK343
DescriptionA potent histone H3-lysine 27 (H3K27) methyltransferase EZH2 inhibitor (IC50 = 4 nM). Diplays 1000-fold selectivity for other HMTs except EZH1 (60-fold selectivity). GSK343 inhibits H3K27 methylation in HCC1806 cells with an IC50 of <200nM (measured by immunofluorescence). MW: 541.69. Purity ≥99% by HPLC
Size5 mg
Concentrationn/a
Applicationsn/a
Other Names1-Isopropyl-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-6-(2-(4-methylpiperazin-1-yl)pyridine-4-yl)-1H-indazole-4-carboxamide
Gene, Accession, CAS #n/a
Catalog #2281-5
Price
Order / More InfoGSK343 from BIOVISION, INC.
Product Specific Referencesn/a
產(chǎn)品資料
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