產(chǎn)品名稱 EPZ 015666 from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 6516/25
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 25 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
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Product NameEPZ 015666
DescriptionPotent and selective protein arginine methyltransferase 5 (PRMT5) inhibitor (IC50 = 22 nM, Ki = 5 nM). Displays selectivity for PRMT5 over a panel of 20 other protein methyltransferases. Exhibits dose-dependent antitumor effects in multiple mantle cell lymphoma (MCL) xenograft models. Orally bioavailable. Purity 98%. MW (observed): 383.44
Size25 mg
Concentrationn/a
Applicationsn/a
Other NamesN-[(2S)-3-(3,4-Dihydro-2(1H)-isoquinolinyl)-2-hydroxypropyl]-6-(3-oxetanylamino)-4-pyrimidinecarboxamide
Gene, Accession, CAS #CAS: 1616391-65-1
Catalog #6516/25
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Order / More InfoEPZ 015666 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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