產(chǎn)品名稱 MJ15 from CAYMAN CHEMICAL COMPANY
產(chǎn)品貨號(hào) 11956-5
產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
產(chǎn)品規(guī)格 5 mg
產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
產(chǎn)品概述
產(chǎn)品詳情
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Product NameMJ15
DescriptionA potent CB1 receptor antagonist (IC50 = 118.9 pM; Ki = 27.2 pM for rat CB1); selective for CB1 over CB2, exhibiting only 46% inhibition of CB2 at a concentration of 10 μM; reverses (+)-WIN 55,212-2 inhibition of forskolin-induced cAMP accumulation in a dose-dependent manner in CHO cells expressing human CB1; reduces food intake and body weight gain in a rat model of diet-induced obesity at a dose of 40 mg/kg; reduces body weight gain and white adipose accumulation in a mouse model of early onset diet-induced obesity
Size5 mg
Concentrationn/a
Applicationsn/a
Other NamesMJ-15 CB-1
Gene, Accession, CAS #CAS: 944154-76-1
Catalog #11956-5
Price
Order / More InfoMJ15 from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
產(chǎn)品資料
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