產(chǎn)品名稱(chēng) AZ Dyrk1B 33 from TOCRIS BIOSCIENCE
產(chǎn)品貨號(hào) 5632/10
產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話(huà):010-67529703
產(chǎn)品規(guī)格 10 mg
產(chǎn)品品牌 TOCRIS BIOSCIENCE
產(chǎn)品概述
產(chǎn)品詳情
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Product NameAZ Dyrk1B 33
DescriptionPotent and selective ATP-competitive Dyrk1B kinase inhibitor (IC50 = 7 nM); displays distinct cellular effects when compared to DYRK1B knockdown through siRNA. Demonstrates cellular in vitro activity (IC50 = 194 nM). Exhibits better selectivity than AZ 191 (Cat. No 5232); displays no off-target effects against a panel of 124 kinases tested (no kinase was inhibited above 50% at 1 μM). Purity 98%. MW (observed): 300.36
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine
Gene, Accession, CAS #CAS: 1679330-37-0
Catalog #5632/10
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Order / More InfoAZ Dyrk1B 33 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
產(chǎn)品資料
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